Bioorganic and Medicinal Chemistry p. 3447 - 3455 (2016)
Update date:2022-08-03
Topics:
Yoshikawa, Masato
Hitaka, Takenori
Hasui, Tomoaki
Fushimi, Makoto
Kunitomo, Jun
Kokubo, Hironori
Oki, Hideyuki
Nakashima, Kosuke
Taniguchi, Takahiko
Utilizing structure-based drug design techniques, we designed and synthesized phosphodiesterase 10A (PDE10A) inhibitors based on pyridazin-4(1H)-one. These compounds can interact with Tyr683 in the PDE10A selectivity pocket. Pyridazin-4(1H)-one derivative
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