Journal of Medicinal Chemistry p. 3290 - 3294 (1991)
Update date:2022-09-26
Topics:
Suto
Stier
Winters
Turner
Pinter
Elliott
Sebolt-Leopold
A series of 3,5-disubstituted-2,1-benzisoxazole-4,7-diones was synthesized and evaluated as radiosensitizers both in vitro and in vivo. These compounds were designed as non-nitro electron-affinic agents in an effort to alleviate some of the toxicities see
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