α-Azido Acids in Heterocyclic Synthesis

DOI: 10.1016/0040-4039(91)80066-F

Source and publish data:

Tetrahedron Letters p. 5493 - 5496 (1991)

Update date:2022-08-05

Topics:

Authors:

Goldstein, Steven W.

McDermott, Ruth E.

Makowski, Michael R.

Eller, Cynthia

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(91)80066-F

2-Aminobenzophenones and acetophenones were N-acylated with α-azido carboxylic acids to give the corresponding anilides.Reductive cyclization provided 3-substituted-2H-1,4-benzodiazepin-2-ones in good (46-99percent) yields.

Full text of DOI:10.1016/0040-4039(91)80066-F

Products guided by the article

Product name:2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-7,8-dimethoxy-5-methyl-3-pentyl-

Cas No:137959-53-6

R&D Labs maybe for 137959-53-6

Chengdu Gelipu Biotechnology Co., Ltd.

website:http://www.glp-china.com

Contact:86-28-82610909

Address:chegndu
Shandong Yubin Chemical CO.,LTD

website:http://www.yukaichem.com/en.html

Contact:+86-536-8865336

Address:binhai economic development zone，262737 shangdong，china
ShenZhen InnoSyn Biotech Co.,Ltd

website:http://www.innosyns.com

Contact:+86-755-28351685

Address:Floor 5 & 6, Building A1, HAIKEXING Strategic Innovative Industrial Park, 16 BaoShan Road, PingShan District
FOSHAN NANHAI ZHONGNAN PHARMACEUTICAL FACTORY

Contact:0086-0757-85609331

Address:XIAHENGTIAN INDUSTRIAL ZONE,SHAYONG VILLAGE,LISHUI TOWN
Jewim Pharmaceutical (Shandong) Co., Ltd

Contact:+8615621883869

Address:山东省泰安市高新技术产业开发区配天门大街西首

Relevant to this article

Enantioselective total synthesis and biological evaluation of (+)-kibdelone A and a tetrahydroxanthone analogue

Doi:10.1021/jo401169z
(2013)
Supramolecular [M₄L₄] tetrahedra based on triangular acylhydrazone catechol ligands

Doi:10.1002/ejoc.201101725
(2012)
Rapid, two-pot procedure for the synthesis of dihydropyridinones; total synthesis of aza-goniothalamin

Doi:10.3762/bjoc.16.15
(2020)
TOTAL SYNTHESIS OF A NEW INHIBITOR OF SUPEROXIDE ANION GENERATION, OPC-15161

Doi:10.1016/S0040-4039(00)79453-6
(1991)
Scandium(III)-zeolites as new heterogeneous catalysts for imino-diels-alder reactions

Doi:10.1002/chem.201103624
(2012)
STEREOSELECTIVE CYCLOPROPANATION OF HOMOALLYLIC ALCOHOLS. FORMAL ATTACHMENT OF A CYCLOPROPANE TO A PREEXISTING RING

Doi:10.1016/S0040-4039(00)93542-1
(1991)

Article Doi