N-Methylated Analogs of Ac28,31>CCK(26-33): Synthesis, Activity, and Receptor Selectivity

DOI: 10.1021/jm00093a013

Source and publish data:

Journal of Medicinal Chemistry p. 2806 - 2811 (1992)

Update date:2022-07-29

Topics:

Authors:

Ron, D. Ron, D.

Gilon, C.

Hanani, M.

Vromen, A.

Selinger, Z.

Chorev, M.

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Article abstract of DOI:10.1021/jm00093a013

A series of singularly N-methylated analogs of Ac28,31>CCK(26-33) were synthesized by the solid-phase methodology, and their biological activity was tested in three different in vitro bioassays.The bioassays employed were the guinea pig gal

Full text of DOI:10.1021/jm00093a013

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Product name:AcAsp-Tyr(SO₃^-Na⁺)-Nle-Gly-Trp-Nle-Asp-(N-Me)PheNH₂

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