Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with δ opioid receptor selectivity

DOI: 10.1021/jm00091a006

Source and publish data:

Journal of Medicinal Chemistry p. 2384 - 2391 (1992)

Update date:2022-08-04

Topics:

Authors:

Toth Toth

Russell Russell

Landis Landis

Kramer Kramer

Fang Fang

Knapp Knapp

Davis Davis

Burks Burks

Yamamura

Hruby Hruby

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Article abstract of DOI:10.1021/jm00091a006

The conformationally restricted, cyclic disulfide-containing δ opioid receptor selective enkephalin analogue [D-Pen²,D-Pen⁵]enkephalin (DPDPE) was modified by 2' (CH₃) and 3' (I, OCH₃, NO₂, NH_{2
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Full text of DOI:10.1021/jm00091a006

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