
Tetrahedron Letters p. 4549 - 4552 (1992)
Update date:2022-08-05
Topics:
Peyman, Anusch
Budt, Karl-Heinz
Spanig, Joerg
Stowasser, Bernd
Ruppert, Dieter
The synthesis of the previously not accessible symmetrical bis(α-aminoalkyl)phosphinic acids is demonstrated. These compounds are valuable central building blocks in the synthesis of HIV protease inhibitors.
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