The squalestatins: Synthesis of C-4 carboxamide derivatives

DOI: 10.1016/S0040-4039(96)02049-7

Source and publish data:

Tetrahedron Letters p. 8925 - 8928 (1996)

Update date:2022-08-05

Topics:

Authors:

Chan, Chuen

Scicinski, Jan J.

Srikantha, Anton R. P.

Watson, Nigel S.

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Article abstract of DOI:10.1016/S0040-4039(96)02049-7

Synthesis of squalestatin S1 C-4 carboxamide, 2, as well as related C-4 amides and C-4 hydroxymethyl derivatives possessing a C-3 hydroxymethyl group (15 and 19) together with their SQS inhibitory activities are presented. Copyright (C) 1996 Elsevier Science Ltd.

Full text of DOI:10.1016/S0040-4039(96)02049-7

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