Synthesis of enantiomerically pure 6,10-epoxybenzocycloocten-7-amines with CNS-activity

DOI: 10.1002/ardp.19923251110

Source and publish data:

Archiv der Pharmazie p. 733 - 739 (1992)

Update date:2022-07-29

Topics:

Authors:

Wunsch Wunsch

Zott Zott

Hofner Hofner

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ardp.19923251110

In an oxa-Pictet-Spengler reaction the methyl (S)-phenyllactate 6 and methyl levulinate (7a) are condensed to the 2-benzopyrans cis-8a and trans-8a, which react with CH₃I to yield the dimethyl ethers cis-9a and trans-9a. Cis-9a and trans-9a can

Full text of DOI:10.1002/ardp.19923251110

Products guided by the article

Product name:Menthyl-5,9-epoxy-5,6,9,10-tetrahydro-8-hydroxy-2,3-dimethoxy-5-methyl-benzocycloocten-7-carboxylat

Cas No:145653-74-3

R&D Labs maybe for 145653-74-3

Jiangxi Hito Chemical Co., Ltd.

Contact:+86-792-3170318

Address:No. 6, Tianhong Ave., Xinghuo Industry Park, Yongxiu, Jiujiang, Jiangxi, China
ZHIJIANG ZENVA SINO COMMERCE AND TRADE CO., LTD.

website:http://www.zenvasino.com

Contact:+86-138-72658998

Address:Shibeishan Road,Zhijiang, Hubei, China
XZL BIO-TECHNOLOGY CO., LTD.

Contact:0086 533 2282832

Address:Zibo，Shandong
MTT Pharma & Bio-technology Co.,Ltd(expird)

Contact:+86-21-58407925

Address:Room2019, Building C, Tomson Center, No.158, Zhang Yang Road, Shanghai, China
Shanghai Korey Pharm Co.,Ltd.(expird)

Contact:021-61840961 021-61840962

Address:No.157,Zhuguang Rd, Qingpu, Shanghai, China

Relevant to this article

Stibine-protected Au₁₃ nanoclusters: Syntheses, properties and facile conversion to GSH-protected Au₂₅ nanocluster

Doi:10.1039/c8sc03132k
(2018)
N-NITROSOHYDROXYLAMINES I. ACETOLYSIS AND ACID-CATALYZED HYDROLYSIS OF N,O-DIBENZYL-N-NITROSOHYDROXYLAMINES. REACTION WITH POTASSIUM t-BUTOXIDE

Doi:10.1016/S0040-4020(01)89037-2
(1992)
Synthesis of Phosphonic Acid Derivatives by Oxidative Activation of Phosphinate Esters

Doi:10.1021/jo00254a015
(1988)
Lewis Acid-Catalyzed Nitrone Cycloadditions to Bidentate and Tridentate α,β-Unsaturated Ketones. High Rate Acceleration, Absolutely endo-Selective and Regioselective Reactions

Doi:10.1016/S0040-4039(00)74770-8
(1992)
Discovery of ANT3310, a Novel Broad-Spectrum Serine β-Lactamase Inhibitor of the Diazabicyclooctane Class, Which Strongly Potentiates Meropenem Activity against Carbapenem-Resistant Enterobacterales and Acinetobacter baumannii

Doi:10.1021/acs.jmedchem.0c01535
(2020)
Dioxygen-triggered transannular dearomatization of benzo[5]helicene diols: Highly efficient synthesis of chiral π-extended diones

Doi:10.1002/anie.201400486
(2014)

Article Doi