Journal of Medicinal Chemistry p. 1319 - 1323 (1993)
Update date:2022-08-03
Topics:
Gerzon, Koert
Humerickhouse, Rod A.
Besch, Henry R.
Bidasee, Keshore R.
Emmick, Jeffrey T.
et al.
Amino- and guanidinoacyl esters of ryanodine were prepared to evaluate the effect of basicity on the binding affinity of these derivatives for the sarcoplasmic reticulum Ca2+-release channel (SR CRC). In the presence of DCC and DMAP Cbz-β-alani
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