Synthesis and inhibitory activities against enkephalin degrading aminopeptidase of H-Trp(Nps)-Lys-OMe analogues bearing chelating groups.

DOI: 10.1002/ardp.19923251202

Source and publish data:

Archiv der Pharmazie p. 743 - 749 (1992)

Update date:2022-08-04

Topics:

Authors:

Gonzalez-Muniz

Harto Harto

de Ceballos

del Rio del Rio

Garcia-Lopez

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Article abstract of DOI:10.1002/ardp.19923251202

With the aim of increasing the inhibitory potency of the analgesic dipeptide H-Trp(Nps)-Lys-OMe against enkephalin-degrading aminopeptidases, the following derivatives bearing chelating groups at the N-terminus have been synthesized: Ac-Trp(Nps)-Lys-OMe (

Full text of DOI:10.1002/ardp.19923251202

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Product name:Trp(Nps)-Lys(Z)-OMe*HCl

Cas No:146791-85-7

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