Synthesis and inhibitory activities against enkephalin degrading aminopeptidase of H-Trp(Nps)-Lys-OMe analogues bearing chelating groups.

DOI: 10.1002/ardp.19923251202

Source and publish data:

Archiv der Pharmazie p. 743 - 749 (1992)

Update date:2022-08-04

Topics:

Authors:

Gonzalez-Muniz

Harto Harto

de Ceballos

del Rio del Rio

Garcia-Lopez

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Article abstract of DOI:10.1002/ardp.19923251202

With the aim of increasing the inhibitory potency of the analgesic dipeptide H-Trp(Nps)-Lys-OMe against enkephalin-degrading aminopeptidases, the following derivatives bearing chelating groups at the N-terminus have been synthesized: Ac-Trp(Nps)-Lys-OMe (

Full text of DOI:10.1002/ardp.19923251202

Products guided by the article

Product name:Trp(Nps)-Lys(Z)-OMe*HCl

Cas No:146791-85-7

R&D Labs maybe for 146791-85-7

Zhengzhou Institute of Chiral Pharmer Research Co., Ltd.

Contact:86-371-55219111

Address:15 Floor, 2 Building, Central China Technovalley, Zhongyuan West Road
Zhushan County Tianxin Pharmaceutical & Chemical Co., Ltd.

Contact:0086-719-4224892

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Hangzhou Gangjin Chemical Co.,Ltd.(expird)

Contact:+86-571-85109780

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ZHEJIANG JIANYE CHEMICAL CO.,LTD.

Contact:86-571-64149273,64149234

Address:No. 48, Fuxi Road, Meicheng Town
Anhui Jiatiansen Agrochemical Co.,Ltd

Contact:15366811918

Address:chemical industrial park,xiangyu town,dongzhi county,anhui,china

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