Synthesis and inhibitory activities against enkephalin degrading aminopeptidase of H-Trp(Nps)-Lys-OMe analogues bearing chelating groups.

DOI: 10.1002/ardp.19923251202

Source and publish data:

Archiv der Pharmazie p. 743 - 749 (1992)

Update date:2022-08-04

Topics:

Authors:

Gonzalez-Muniz

Harto Harto

de Ceballos

del Rio del Rio

Garcia-Lopez

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ardp.19923251202

With the aim of increasing the inhibitory potency of the analgesic dipeptide H-Trp(Nps)-Lys-OMe against enkephalin-degrading aminopeptidases, the following derivatives bearing chelating groups at the N-terminus have been synthesized: Ac-Trp(Nps)-Lys-OMe (

Full text of DOI:10.1002/ardp.19923251202

Products guided by the article

Product name:Trp(Nps)-Lys(Z)-OMe*HCl

Cas No:146791-85-7

R&D Labs maybe for 146791-85-7

Chengdu Baishixing Science and Technology Industry Co., Ltd.

website:http://www.cd-bsx.com

Contact:+86-28-88531548

Address:#217,North of Industry Road,Heshan Town,Pujiang County,Chengdu,Sichuan,China.
Shandong Jiulong Hisince Pharmaceutical Co.,Ltd.

Contact:+86-15853188990

Address:Huadian Pioneer Park, Huadian Township, Qihe County, Dezhou City, Shandong, P.R.China
Onlychem (Jinan)Biotech Co.,Ltd

Contact:86-531-83175885

Address:No. 44, Honglou South Road, Jinan,China
Wuhan Silworld Chemical Co.,Ltd

website:http://www.silworldchemical.com

Contact:+86-27-85613400

Address:No.198 jiangjun Road, Wuhan,China 430033
New Forms

Contact:+31-24-3886056

Address:Binderskampweg 29 Unit 36

Relevant to this article

Concerning the reaction mechanism of the hydantoin synthesis according to Biltz, II: Influence of substituents on the direction of the rearrangement

Doi:10.1002/ardp.19933260110
(1993)
Enantioselective synthesis of optically active secondary amines via asymmetric reduction

Doi:10.1016/S0957-4166(00)86063-2
(1992)
Alkynyl sulfides and selenides from alkynyl bromides and diorganoyl chalcogenides promoted by copper(I) iodide

Doi:10.1016/0040-4039(93)85084-A
(1993)
Comparison of Conventional and Microwave Assisted Reactions Giving Aromatic Oxazolidines

Doi:10.1007/s00706-003-0020-6
(2003)
Organocatalyzed direct glycosylation of unprotected and unactivated carbohydrates

Doi:10.1021/ol402914v
(2013)
Exploration of the expeditious potential of Pseudomonas fluorescens lipase in the kinetic resolution of racemic intermediates and its validation through molecular docking

Doi:10.1002/chir.22771
(2018)

Article Doi