Synthesis and inhibitory activities against enkephalin degrading aminopeptidase of H-Trp(Nps)-Lys-OMe analogues bearing chelating groups.

DOI: 10.1002/ardp.19923251202

Source and publish data:

Archiv der Pharmazie p. 743 - 749 (1992)

Update date:2022-08-04

Topics:

Authors:

Gonzalez-Muniz

Harto Harto

de Ceballos

del Rio del Rio

Garcia-Lopez

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Article abstract of DOI:10.1002/ardp.19923251202

With the aim of increasing the inhibitory potency of the analgesic dipeptide H-Trp(Nps)-Lys-OMe against enkephalin-degrading aminopeptidases, the following derivatives bearing chelating groups at the N-terminus have been synthesized: Ac-Trp(Nps)-Lys-OMe (

Full text of DOI:10.1002/ardp.19923251202

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Product name:Trp(Nps)-Lys(Z)-OMe*HCl

Cas No:146791-85-7

R&D Labs maybe for 146791-85-7

Hubei Xinghuo Chemical Co., Ltd.,

Contact:13925817279 13907299441

Address:Xinghuo Fine Chemistry Industrial Park, Xiaochang County, Hubei Province, China
Landz International Company Ltd.

Contact:0086-21-58891610

Address:985 Dongfang Road, Pudong, Shanghai 200122 China
Shanxi Sanwei Group Co.,Ltd

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Address:Zhaocheng town, Hongtong County, Linfen City, Shanxi Province
ZhangJiaGang YaRui Chemical Co.,Ltd.

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Address:China JiangSu Province Zhang Jia Gang City YangShe Oriental Plaza Building 10 B307
Changzhou BaoKang Pharmaceutical & Chemical Co., Ltd

Contact:(86) 519-88782201 88784080 88785278

Address:Henglin town, changzhou,Jiangsu

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