Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: Structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4- [3-[(1-methylethyl)amino]-pyridinyl]piperazine monomethanesulfonate (U- 90152S), a second-generation clinical candidate

DOI: 10.1021/jm00062a027

Source and publish data:

Journal of Medicinal Chemistry p. 1505 - 1508 (1993)

Update date:2022-07-31

Topics:

Authors:

Romero

Morge

Genin

Biles

Busso

Resnick

Althaus

Reusser

Thomas

Tarpley