Lactones, XXIII: Synthesis and stereochemistry of 'γ-lactonized' butyrophenone-type neuroleptics

DOI: 10.1002/ardp.19933260111

Source and publish data:

Archiv der Pharmazie p. 51 - 55 (1993)

Update date:2022-08-04

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Authors:

Lehmann Lehmann

Radwansky

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Article abstract of DOI:10.1002/ardp.19933260111

'γ-Lactonized' neuroleptics (1,2a-c) can be obtained by reaction of α-formyl, α-carboxy- and α-methylene-lactones 5-7a,b with amines 8a-c. 6a, 1a-c were cis/trans-mixtures with predominating cis-compounds, 6b, 2a cis/trans-mixtures with predominating tran

Full text of DOI:10.1002/ardp.19933260111

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