Studies on aromatase inhibitors. I. Synthesis and biological evaluation of 4-amino-4H-1,2,4-triazole derivatives

DOI: 10.1248/cpb.44.1871

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1871 - 1879 (1996)

Update date:2022-08-04

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Authors:

Okada, Minoru

Yoden, Toru

Kawaminami, Eiji

Shimada, Yoshiaki

Kudoh, Masafumi

Isomura, Yasuo

Shikama, Hisataka

Fujikura, Takashi

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Article abstract of DOI:10.1248/cpb.44.1871

Various 4-N-substituted amino-4H-1,2,4-triazole derivatives were synthesized and evaluated for aromatase-inhibitory activity (in vitro) and for pregnant mare serum gonadotropin (PMSG)-induced estrogen synthesis- inhibitory activity (in vivo). The 4-(4-cya

Full text of DOI:10.1248/cpb.44.1871

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Product name:4-[N-acetyl-N-(4-nitrophenyl)amino]-4H-1,2,4-triazole

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