Chemical and Pharmaceutical Bulletin p. 1871 - 1879 (1996)
Update date:2022-08-04
Topics:
Okada, Minoru
Yoden, Toru
Kawaminami, Eiji
Shimada, Yoshiaki
Kudoh, Masafumi
Isomura, Yasuo
Shikama, Hisataka
Fujikura, Takashi
Various 4-N-substituted amino-4H-1,2,4-triazole derivatives were synthesized and evaluated for aromatase-inhibitory activity (in vitro) and for pregnant mare serum gonadotropin (PMSG)-induced estrogen synthesis- inhibitory activity (in vivo). The 4-(4-cya
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