Adenosine receptor prodrugs: Synthesis and biological activity of derivatives of potent, A1-selective agonists

DOI: 10.1002/jps.2600830112

Source and publish data:

Journal of Pharmaceutical Sciences p. 46 - 53 (1994)

Update date:2022-08-05

Topics:

Authors:

Maillard

Nikodijevic

LaNoue LaNoue

Berkich Berkich

Bartus Bartus

Jacobson

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Article abstract of DOI:10.1002/jps.2600830112

5'-Ester derivatives of the potent adenosine agonists N⁶-[4-[[[[4-[[[(2- acetylaminoethyl)amino]carbonyl]methyl]anilino]carbonyl]methyl]phenyl]adenosi ne (N-AcADAC; 1) and N⁶-cyclopentyladenosine (CPA; 2) were prepared as prodrugs. B

Full text of DOI:10.1002/jps.2600830112

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