2-Substituted 5-methoxy-N-acyltryptamines: Synthesis, binding affinity for the melatonin receptor, and evaluation of the biological activity

DOI: 10.1021/jm00077a010

Source and publish data:

Journal of Medicinal Chemistry p. 4069 - 4074 (1993)

Update date:2022-08-04

Topics:

Authors:

Spadoni Spadoni

Stankov Stankov

Duranti Duranti

Biella Biella

Lucini Lucini

Salvatori

Fraschini

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Article abstract of DOI:10.1021/jm00077a010

A series of 2-substituted 5-methoxy-N-acyltryptamines was synthesized and their affinity for the melatonin receptor, isolated from whole quail brains, was tested in a succession of in vitro ligand-receptor binding experiments, using 2-[¹²⁵I]iod

Full text of DOI:10.1021/jm00077a010

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