
Journal of Heterocyclic Chemistry p. 1357 - 1359 (1993)
Update date:2022-09-26
Topics:
Cignarella
Villa
Barlocco
A new series of 8-substituted-2,8-diazaspiro[4.5]decan-3-ones has been synthesized and tested in in vitro and in vivo assays predictive for cholinergic activity, in comparison with the muscarinic agent RS-86. Preliminary pharmacological data indicate that
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