
Journal of Medicinal Chemistry p. 2552 - 2563 (1994)
Update date:2022-08-03
Topics:
Norman, Mark H.
Rigdon, Greg C.
Navas, Frank
Cooper, Barrett R.
A series of novel 4-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)butyl cyclic amides was prepared and evaluated as potential antipsychotic agents. The target compounds were examined in vitro for their binding affinities to the dopamine D2, serotonin 5-HT2,
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Doi:10.1021/jacs.5b03017
(2015)Doi:10.1002/anie.201811859
(2019)Doi:10.1021/acscatal.9b02461
(2019)Doi:10.1002/anie.202002258
()Doi:10.1016/0022-1139(93)02956-F
(1994)Doi:10.1055/s-1997-1499
(1997)