Palladium-Catalyzed Heteroarylation of 1-(tert-Butyldimethylsilyl)-3-indolylzinc Chloride. Efficient Synthesis of 3-(2-Pyridyl)indoles

DOI: 10.1016/S0040-4039(00)75819-9

Source and publish data:

Tetrahedron Letters p. 793 - 796 (1994)

Update date:2022-08-05

Topics:

Authors:

Amat, Mercedes

Hadida, Sabine

Bosch, Joan

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)75819-9

Palladium-catalyzed coupling of 1-(tert-butyldimethylsilyl)-3-indolylzinc chloride (2) with either ?-deficient or ?-excedent heteroaryl halides gives 3-arylindoles in good to excellent yields.The method is extensively applied to the preparation of 3-(2-pyridyl)indoles.

Full text of DOI:10.1016/S0040-4039(00)75819-9

Products guided by the article

Product name:1-(benzenesulfonyl)-1'-(tert-butyldimethylsilyl)-3,3'-biindole

Cas No:155440-55-4

R&D Labs maybe for 155440-55-4

Shanghai Bojing Chemical Co., Ltd.

Contact:021-37122233

Address:6F Buildiing 11,No.388,Baifu Road,District Fengxian.Shanghai, China.
Guilin Zhenda Bio-Tech Co., Ltd.

Contact:86-773-3568977

Address:-Yangtang shangshui industry park, Lingui county,
NEWSTAR CHEM ENTERPRISE LTD.

Contact:0572-2722882

Address:1201,F3,xinghuibandao,
JiYi Chemical (Beijing) Co., Ltd.

Contact:+86-10-89385733

Address:Shilou Town of Fangshan District， Beijing
Innua Petrochem Ltd.

Contact:+1-284-4950244

Address:Box 3069, Road Town, Tortola, British Virgin Islands

Relevant to this article

Cocaine and 3β-(4'-substituted phenyl)tropane-2β-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter

Doi:10.1021/jm00002a020
(1995)
A novel synthesis of quinazolinequinone and carbazolequinone through anionic cycloaddition: Its application to a synthesis of murrayaquinone A

Doi:10.1248/cpb.42.416
(1994)
Design and synthesis of a new class of nonmacrocyclic alkali metal host compounds

Doi:10.1021/ol006468o
(2000)
Oxidative catalysis using the stoichiometric oxidant as a reagent: An efficient strategy for single-electron-transfer-induced tandem anion-radical reactions

Doi:10.1002/anie.201403776
(2014)
RING-TRANSFORMATION EQUILIBRIUM WITH PARTICIPATION OF ?-BONDED S(IV) IN AN ISOTHIAZOLE SYSTEM. SYNTHESIS OF NON-RING-TRANSFORMED 5-(2-AMINOVINYL)ISOTHIAZOLE DERIVATIVE VIA 1,3-SILYL GROUP SHIFT

Doi:10.1016/S0040-4039(01)81493-3
(1984)
Magnetostructural correlation in tetracopper(II) cubanes

Doi:10.1016/j.poly.2013.12.010
(2014)

Article Doi