Journal of Enzyme Inhibition and Medicinal Chemistry p. 124 - 131 (2014)
Update date:2022-08-05
Topics:
Zubriene, Asta
Capkauskaite, Edita
Gylyte, Joana
Kisonaite, Migle
Tumkevicius, Sigitas
Matulis, Daumantas
A series of benzenesulfonamide derivatives, bearing benzimidazole moieties, were designed and synthesized as inhibitors of carbonic anhydrases (CAs). Their binding affinities to recombinant human CA isozymes I, II, VII, XII and XIII were determined by the
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