Synthesis of (S)-3,4-diaminobutanenitriles as precursors for 3-amino-GABA derivatives

DOI: 10.1002/ardp.19953280311

Source and publish data:

Archiv der Pharmazie p. 265 - 268 (1995)

Update date:2022-08-06

Topics:

Authors:

Gmeiner Gmeiner

Hummel Hummel

Haubmann

Hofner Hofner

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Article abstract of DOI:10.1002/ardp.19953280311

Starting from natural asparagine (1) a synthesis of the protected (S)-3,4-diaminobutanenitriles 5 and 8a-c via the β-homoserine derivative 2 is described. The amino function in position 4 was introduced by Mitsunobu-coupling or by reductive amination when

Full text of DOI:10.1002/ardp.19953280311

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