Studies on pyridonecarboxylic acids. III. Synthesis and antibacterial activity evaluation of 1,8-disubstituted 6-fluoro-4-oxo-7-piperazinyl-4H-[1,3]thiazeto[3,2-a] quinoline-3-carboxylic acid derivatives

DOI: 10.1248/cpb.43.63

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 63 - 70 (1995)

Update date:2022-08-02

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Authors:

Segawa Segawa

Kazuno Kazuno

Matsuoka

Shirahase

Ozaki Ozaki

Matsuda Matsuda

Tomii Tomii

Kitano Kitano

Kise Kise

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Article abstract of DOI:10.1248/cpb.43.63

A series of 1,8-disubstituted 6-fluoro-4-oxo-7-piperazinyl-4H-[1,3]thiazeto[3,2-a] quinoline-3-carboxylic acid derivatives was prepared and evaluated for antibacterial activity. In the 7-piperazinyl series, addition of a fluorine at C-8, which increased t

Full text of DOI:10.1248/cpb.43.63

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