Synthesis of 7-, 8- and 9-Membered Rings via endo Heck Cyclisations of Amino Acid Derived Substrates

DOI: 10.1039/C39950001743

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 1743 - 1744 (1995)

Update date:2022-08-04

Topics:

Authors:

Gibson, Susan E.

Middleton, Richard J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1039/C39950001743

Aryl iodides tethered to dehydroalanine units by two to four methylene groups undergo intramolecular Heck reactions under anhydrous Jeffery conditions to give 7-, 8- and 9-membered rings by the endo-mode of cyclisation; under harsher conditions, a palladi

Full text of DOI:10.1039/C39950001743

View Article Online / Journal Homepage / Table of Contents for this issue

View Article Online

Products guided by the article

Product name:2-{Acetyl-[2-(2-iodo-phenyl)-ethyl]-amino}-acrylic acid methyl ester

Cas No:171734-15-9

R&D Labs maybe for 171734-15-9

Beijing Top Science biological technology co., LTD

Contact:+86-13439059536

Address:15-1705 jre three mile, Beijing 100000,CHINA
HANGZHOU ZHONGCHANG SCIENTIFIC CO.,LTD

Contact:+86-571-88932183

Address:Hangzhou
FOSHAN NANHAI ZHONGNAN PHARMACEUTICAL FACTORY

Contact:0086-0757-85609331

Address:XIAHENGTIAN INDUSTRIAL ZONE,SHAYONG VILLAGE,LISHUI TOWN
Tianjin Jiuri New Materials Co., Ltd.

Contact:+86-22-58889220

Address:C-5/6, Vison Hill, No.1 Gonghua Road, Huayuan Hi-tech Park, Tianjin, China.
QUZHOU ZIO I/E CO.;LTD

Contact:13357117572

Address:No.149 Shiji dadao Road.

Relevant to this article

Effective nitration of anilides and acrylamides by tert-butyl nitrite

Doi:10.1002/ejoc.201403510
(2015)
A facile one-pot synthesis of 3,5-disubstituted isoxazole derivatives using hydroxy (tosyloxy) iodobenzene

Doi:10.1002/jhet.1556
(2013)
QUANTITATIVE SEPARATION AND ANALYSIS OF DIASTEREOMERS OF L-METHIONINE-S,R-SULFOXIMINE VIA CYCLIC N-BLOCKED DERIVATIVES

Doi:10.1016/S0040-4039(00)81684-6
(1983)
A total synthesis of grifolin

Doi:10.1248/cpb.36.2239
(1988)
Synthesis and some chemical transformations of N-cyclohexyl-2-imino-4- methyl-5,5-pentamethylene-2,5-dihydrofuran-3-carboxamide

Doi:10.1134/S1070428009100303
(2009)
1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A₂α and fatty acid amide hydrolase

Doi:10.1016/j.bmc.2009.11.028
(2010)

Article Doi