Journal of Medicinal Chemistry
Page 28 of 30
1
2
3
4
5
6
7
8
9
16.
Matthews, J. E.; Jansen, M.; Lyerly, D.; Cox, R.; Chen, W.-J.; Koller, K. J.; Daniels, A. J.
Pharmacological characterization and selectivity of the NPY antagonist GR231118
(1229U91) for different NPY receptors. Regul. Pept. 1997, 72, 113-119.
17.
Schober, D. A.; Gackenheimer, S. L.; Heiman, M. L.; Gehlert, D. R. Pharmacological
characterization of 125I-1229U91 binding to Y1 and Y4 neuropeptide Y/peptide YY
receptors. J. Pharmacol. Exp. Ther. 2000, 293, 275-280.
18.
Balasubramaniam, A.; Mullins, D. E.; Lin, S.; Zhai, W.; Tao, Z.; Dhawan, V. C.; Guzzi,
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
M.; Knittel, J. J.; Slack, K.; Herzog, H.; Parker, E. M. Neuropeptide Y (NPY) Y4 receptor
selective agonists based on NPY(32−36):ꢀ development of an anorectic Y4 receptor
selective agonist with picomolar affinity. J. Med. Chem. 2006, 49, 2661-2665.
19.
Li, J.-B.; Asakawa, A.; Terashi, M.; Cheng, K.; Chaolu, H.; Zoshiki, T.; Ushikai, M.;
Sheriff, S.; Balasubramaniam, A.; Inui, A. Regulatory effects of Y4 receptor agonist (BVD-
74D) on food intake. Peptides 2010, 31, 1706-1710.
20.
Robinson, A. J.; Elaridi, J.; Van Lierop, B. J.; Mujcinovic, S.; Jackson, W. R.
Microwave-assisted RCM for the synthesis of carbocyclic peptides. J. Pept. Sci. 2007, 13,
280-285.
21.
metathesis in peptides - the sting is in the tail! Aust. J. Chem. 2011, 64, 806-811.
22. Elaridi, J.; Patel, J.; Jackson, W. R.; Robinson, A. J. Controlled synthesis of (S,S)-2,7-
Van Lierop, B. J.; Bornschein, C.; Jackson, W. R.; Robinson, A. J. Ring-closing
diaminosuberic acid:ꢀ a method for regioselective construction of dicarba analogues of
multicystine-containing peptides. J. Org. Chem. 2006, 71, 7538-7545.
23.
Passarella, D.; Peretto, B.; Blasco y Yepes, R.; Cappelletti, G.; Cartelli, D.; Ronchi,
C.; Snaith, J.; Fontana, G.; Danieli, B.; Borlak, J. Synthesis and biological evaluation of
novel thiocolchicine–podophyllotoxin conjugates. Eur. J. Med. Chem. 2010, 45, 219-226.
24.
diaminopimelic acid via olefin cross-metathesis. Synth. Commun. 2006, 36, 1707-1713.
25. Ward, M. D.; Zhu, Z. Compounds as L-cystine crystallization inhibitors and uses
thereof. US 2012/0316236, Dec.13, 2012, 2012.
26. Hiebl, J.; Blanka, M.; Guttman, A.; Kollmann, H.; Leitner, K.; Mayrhofer, G.;
Nolen, E. G.; Fedorka, C. J.; Blicher, B. Synthesis of orthogonally protected S,S-2,6-
Rovenszky, F.; Winkler, K. A detailed investigation of the preparation of 2,7-
diaminosuberic acid and 2,5-diaminoadipic acid derivatives using Kolbe electrolysis.
Tetrahedron 1998, 54, 2059-2074.
27.
Williams, R. M.; Liu, J. Asymmetric synthesis of differentially protected 2,7-
diaminosuberic acid, a ring-closure metathesis approach. J. Org. Chem. 1998, 63, 2130-
2132.
28.
Aguilera, B.; Wolf, L. B.; Nieczypor, P.; Rutjes, F. P. J. T.; Overkleeft, H. S.; van Hest,
J. C. M.; Schoemaker, H. E.; Wang, B.; Mol, J. C.; Furstner, A.; Overhand, M.; van der Marel,
G. A.; van Boom, J. H. Synthesis of diaminosuberic acid derivatives via ring-closing
alkyne metathesis. J Org Chem 2001, 66, 3584-3589.
29.
Hiebl, J.; Kollmann, H.; Rovenszky, F.; Winkler, K. One step synthesis of
orthogonally protected diaminodicarboxylic acids by mixed kolbe electrolysis. Bioorg.
Med. Chem. Lett. 1997, 7, 2963-2966.
30.
Cabrele, C.; Langer, M.; Beck-Sickinger, A. G. Amino acid side chain attachment
approach and its application to the synthesis of tyrosine-containing cyclic peptides. J.
Org. Chem. 1999, 64, 4353-4361.
31.
Rizzi, L.; Cendic, K.; Vaiana, N.; Romeo, S. Alcohols immobilization onto 2-
chlorotritylchloride resin under microwave irradiation. Tetrahedron Lett. 2011, 52,
2808-2811.
28
ACS Paragon Plus Environment