Total synthesis of deacetyl-caloporoside, a novel inhibitor of the GABA(A) receptor ion channel

DOI: 10.1016/0040-4039(96)00316-4

Source and publish data:

Tetrahedron Letters p. 2453 - 2456 (1996)

Update date:2022-08-04

Topics:

Authors:

Tatsuta Tatsuta

Yasuda Yasuda

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Article abstract of DOI:10.1016/0040-4039(96)00316-4

The total synthesis of deacetyl-caloporoside (1) which contains a β-D-mannopyranoside unit has been accomplished by coupling of the disaccharide-like segment derived from methyl α-D-mannopyranoside, with the hydroxyheptadecyl salicylic acid segment. The biological activity of 1 has also been evaluated.

Full text of DOI:10.1016/0040-4039(96)00316-4

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