Synthesis and pharmacological activity of philanthotoxin-343 analogs: Antagonists of ionotropic glutamate receptors

DOI: 10.1016/S0040-4020(97)00801-6

Source and publish data:

Tetrahedron p. 12391 - 12404 (1997)

Update date:2022-09-26

Topics:

Authors:

Huang, Danwen

Jiang, Hong

Nakanishi, Koji

Usherwood

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Article abstract of DOI:10.1016/S0040-4020(97)00801-6

The synthesis of two classes of Philanthotoxin-343 analogs is described. Quantitative information on the antagonism of quisqualate-sensitive ionotropic glutamate receptors of insect muscle by these compounds is presented.

Full text of DOI:10.1016/S0040-4020(97)00801-6

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