2-Methyl N-(p-toluenesulfinyl)aziridine-2-carboxylic acid: Asymmetric synthesis of α-methylphenylalanine and α-methyl-β-phenylserine

DOI: 10.1016/0040-4039(96)01168-9

Source and publish data:

Tetrahedron Letters p. 5473 - 5476 (1996)

Update date:2022-08-03

Topics:

Authors:

Davis, Franklin A.

Liu, Hu Liu, Hu

Reddy, G. Venkat

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Article abstract of DOI:10.1016/0040-4039(96)01168-9

2-Substituted aziridine 2a, prepared from sulfinimine 1 via a Darzens-type condensation, undergoes a highly regio- and stereocontrolled ring-opening to give α-methylphenylalanine and α-methyl-β-phenylserine in high enantiomeric purity.

Full text of DOI:10.1016/0040-4039(96)01168-9

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