Effective enantioselective approach to α-aminoalkylacrylic acid derivatives via a synthetic equivalent of an asymmetric Baylis-Hillman reaction: Application to the synthesis of two C-2′ hydroxymethyl analogues of docetaxel

DOI: 10.1039/P19960002869

Source and publish data:

Journal of the Chemical Society. Perkin transactions I p. 2869 - 2872 (1996)

Update date:2022-08-04

Topics:

Authors:

Genisson, Yves

Massardier, Christine

Gautier-Luneau, Isabelle

Greene, Andrew E.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1039/P19960002869

Two C-2′ hydroxymethyl analogues of docetaxel have been synthesized from 10-desacetyl baccatin III and enantiopure (3S)-3-(N-tert-butoxycarbonylamino)-2-methylene-3-phenylpropanoic acid; the latter was prepared via the use of a new method, which is discus

Full text of DOI:10.1039/P19960002869

View Article Online / Journal Homepage / Table of Contents for this issue

View Article Online

Products guided by the article

Product name:2-((S)-tert-Butoxycarbonylamino-phenyl-methyl)-acrylic acid (1R,2S)-2-phenyl-cyclohexyl ester

Cas No:186371-33-5

R&D Labs maybe for 186371-33-5

Shanghai Bocimed Pharmaceutical Co., Ltd.

website:http://www.bocimed.com

Contact:+86-21-68861632

Address:Building 1, Lane 647, Songtao Road, Zhangjiang High-Tech Park, Shanghai
SHANGHAI T&W PHARMACEUTICAL CO., LTD.

website:http://www.trustwe.com

Contact:+86-21-61551413

Address:601, No. 1, 2277 Nong, Zu Chongzhi Road, Zhangjiang Hightech. Park, Pudong
Beijing ZhongDaXinHe Chemical Product Co.,Ltd(expird)

Contact:010-52876516

Address:tongzhoubeiyuan
Anhui Asahikasei Chemical Co., Ltd

Contact:86-551-4259770

Address:No. 88 Linquan Road Hefei Anhui China
Changzhou Welton Chemical Co., Ltd,

Contact:0086-519-85910828,85920537,85912897

Address:No.8 Jinlong Road, Binjiang Park, Changzhou, Jiangsu, China.

Relevant to this article

Doi:10.1021/ja00413a068
(1981)
Doi:10.1021/ja01132a021
(1952)
Reactions with Hydrazidoyl Halides XII¹ Synthesis of Pyrazolo[5,1-c]-1,2,4-triazine, Selenadiazolo[3,2-a]quinazolones, Selenadiazoline, Thiadiazoline and Thiazole Derivatives

Doi:10.1002/jccs.199600072
(1996)
Apoptolidin A: Total synthesis and partially glycosylated analogues

Doi:10.1002/chem.200600462
(2006)
Synthesis of a hexasaccharide acceptor corresponding to the reducing terminus of mycobacterial 3-O-methylmannose polysaccharide (MMP)

Doi:10.1016/S0008-6215(96)00239-X
(1996)
Linked benzylamido-cyclopentadienyl ligands: Synthesis and characterization of alkyl titanium complexes

Doi:10.1002/cber.19971300211
(1997)

Article Doi