Zinc-Mediated Allylation of N-Protected α-Amino Aldehydes in Aqueous Solution. Stereoselective Synthesis of Phe-Phe Hydroxyethylene Dipeptide Isosteres

DOI: 10.1055/s-1997-803

Source and publish data:

Synlett p. 351 - 352 (1997)

Update date:2022-08-05

Topics:

Authors:

Hanessian, Stephen

Park, Haeil

Yang, Rui-Yang

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Article abstract of DOI:10.1055/s-1997-803

An efficient route for the synthesis of a Phe-Phe hydroxyethylene dipeptide isostere utilized for the design of potential inhibitors of renin and HIV-protease was developed.

Full text of DOI:10.1055/s-1997-803

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