
Bioorganic and Medicinal Chemistry Letters p. 91 - 96 (1999)
Update date:2022-09-26
Topics:
Imbach, Patricia
Capraro, Hans-Georg
Furet, Pascal
Mett, Helmut
Meyer, Thomas
Zimmermann, Juerg
Novel 2,6,9-substituted purine derivatives represent a class of potent and selective inhibitors of CDK1/cyclinB. The synthesis, SAR and biological profile of selected compounds are described.
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