Novel frameworks for trifluoromethyl ketone and phosphonate TSA inhibitors of type II PLA2

DOI: 10.1016/S0960-894X(97)00246-1

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1421 - 1426 (1997)

Update date:2022-09-26

Topics:

Authors:

Garigipati, Ravi S.

Seibel, George

Mayer, Ruth J.

Bolognese, Brian

McCord, Mark

Marshall, Lisa A.

Adams, Jerry L.

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Article abstract of DOI:10.1016/S0960-894X(97)00246-1

Design and synthesis of some TSA inhibitors on novel molecular frameworks is described. This TSA analog design culminates in the preparation of the phosphonate 18.

Full text of DOI:10.1016/S0960-894X(97)00246-1

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