Synthesis and inhibition analysis of five-membered homoazasugars from D-arabinofuranose via an SN2 reaction of the chloromethylsulfonate

Article abstract of DOI:10.1016/0040-4039(95)01769-E

Five-membered homoazasugars having a side-chain which can be modified to other functional groups or linked to other aglycon moieties were prepared from 2,3,5-tri-O-benzyl-D-arabinofuranose via a favorable SN2 reaction of the chloromethylsulfonate with azi