Tetrahedron Letters p. 4865 - 4868 (1999)
Update date:2022-09-26
Topics:
Piro, Jordi
Rubiralta, Mario
Giralt, Ernest
Diez, Anna
We describe a stereoselective preparation of 3-amino-2-piperidone 1, a new conformationally constrained Ser-Leu surrogate. The key steps of the synthesis of compound I are the lactamisation of the secondary aminolactone 4 and the amination of the 3-position via the sulfite 2.
View MoreContact:+86 755 26588093
Address:No.9 Linkong West Street, Hengdian Street, Huangpi District, Wuhan City, China.
Haitong Chemical Industrial Co.,Ltd.
website:https://www.haitonglongwin.com/
Contact:+86-022-66221018
Address:18-701, No.99, The 4th Street, TEDA,
Chengdu ZY Biochemical Technology Co., LTD
Contact:0086-28-88680086
Address:170 Qingpu Road, Shouan Town, Pujiang County
website:http://www.antimex.com
Contact:0086-21-50563169
Address:Room1027,No.Jinyu Road,Pudong
Zhejiang Rongkai Chemical Technology Co.,Ltd.
Contact:+86-578-8185786
Address:Shangjiang Industrial Zone,Suichang
Doi:10.1021/jm00336a038
(1964)Doi:10.1016/S0040-4020(01)82967-7
(1969)Doi:10.1021/np990089q
(1999)Doi:10.1016/j.tetasy.2004.07.064
(2004)Doi:10.1021/ja01162a101
(1950)Doi:10.1021/ol006465b
(2000)
