Tetrahedron Letters p. 4865 - 4868 (1999)
Update date:2022-09-26
Topics:
Piro, Jordi
Rubiralta, Mario
Giralt, Ernest
Diez, Anna
We describe a stereoselective preparation of 3-amino-2-piperidone 1, a new conformationally constrained Ser-Leu surrogate. The key steps of the synthesis of compound I are the lactamisation of the secondary aminolactone 4 and the amination of the 3-position via the sulfite 2.
View MoreContact:+86-577-65618087-605
Address:Room 402, Unit 4 Xinhu Bldg. Waitan Ruian City, Zhejiang China.
Contact:+86-27-87204219, +86-27-87215023
Address:2402, HuiGu Space-time Building, 8 Forest Road, East Lake Hi-Tech Development Zone
Contact:+86-13666670345
Address:Agricultural Development Zone, Haining, Jiaxing, Zhejiang
Yicheng Goto Pharmaceuticals Co.,Ltd.
Contact:+86 710 3423122
Address:5th Floor,East Gate of Building #2,Servo-Industrial Park,1st Qilin Road,Xiangyang,Hubei,China
Contact:+86-571-86025531 / 86024803
Address:1218-24 Guangyin Mansion,42 Fengqi East Road
Doi:10.1021/jm00336a038
(1964)Doi:10.1016/S0040-4020(01)82967-7
(1969)Doi:10.1021/np990089q
(1999)Doi:10.1016/j.tetasy.2004.07.064
(2004)Doi:10.1021/ja01162a101
(1950)Doi:10.1021/ol006465b
(2000)
