Synthesis and evaluation of isothiocyanate-containing derivatives of the δ-opioid receptor antagonist Tyr-Tic-Phe-Phe (TIPP) as potential affinity labels for δ-opioid receptors

DOI: 10.1021/jm000345s

Source and publish data:

Journal of Medicinal Chemistry p. 5044 - 5049 (2000)

Update date:2022-09-26

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Authors:

Maeda Maeda

Berman Berman

Murray Murray

Aldrich Aldrich

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Article abstract of DOI:10.1021/jm000345s

Derivatives of the δ-opioid receptor-selective peptide antagonist H-Tyr-Tic-Phe-Phe-OH (TIPP) containing an isothiocyanate moiety at the para position of either Phe³ or Phe⁴ were prepared as potential affinity labels for δ-opioid rec

Full text of DOI:10.1021/jm000345s

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