An efficient synthesis of diethyl 1-aminoalkylphosphonate hydrochlorides via the intermediate diethyl 1-azidoalkylphosphonates

Article abstract of DOI:10.1080/00397919208019072

The title compounds 4 have been obtained in high yields in a one-step sequence by the Mitsunobu reaction of diethyl 1-hydroxyalkylphosphonates 1 with hydrazoic acid, and subsequence treatment of the intermediate azides 2 with triphenylphosphine, followed

Full text of DOI:10.1080/00397919208019072

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Synthetic Communications: An
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An Efficient Synthesis
of Diethyl 1-
Aminoalkylphosphonate
Hydrochlorides via the
Intermediate Diethyl 1-
Azidoalkylphosphonates
Tadeusz Gajda a & Maciej Matusiak a
a Institute of Organic Chemistry Technical University,
Zwirki 36, 90-924, Lódź, Poland
Published online: 24 Sep 2006.
To cite this article: Tadeusz Gajda & Maciej Matusiak (1992) An Efficient Synthesis
of Diethyl 1-Aminoalkylphosphonate Hydrochlorides via the Intermediate Diethyl 1-
Azidoalkylphosphonates, Synthetic Communications: An International Journal for
Rapid Communication of Synthetic Organic Chemistry, 22:15, 2193-2203
To link to this article: http://dx.doi.org/10.1080/00397919208019072
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