Bioorganic and Medicinal Chemistry Letters p. 1239 - 1242 (2004)
Update date:2022-07-30
Topics:
Jablonowski, Jill A.
Chai, Wenying
Li, Xiaobing
Rudolph, Dale A.
Murray, William V.
Youngman, Mark A.
Dax, Scott L.
Nepomuceno, Diane
Bonaventure, Pascal
Lovenberg, Timothy W.
Carruthers, Nicholas I.
Through SAR studies of a piperidinylindoline cinnamide HTS lead, the first potent, non-peptide, low molecular weight selective Neuropeptide Y Y 2 (NPY Y2) antagonists have been synthesized. The SAR studies around the piperidinyl, the indolinyl, and the cinnamyl moieties are discussed.
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(1991)Doi:10.1023/A:1015351628312
(2002)Doi:10.1021/ja00871a014
(1962)Doi:10.1002/pola.27708
(2015)Doi:10.1007/BF00901447
(1966)Doi:10.3390/molecules181113588
(2013)