Journal of Medicinal Chemistry p. 2061 - 2064 (2001)
Update date:2022-08-03
Topics:
Brooks
Etgen
Rito
Shuker
Dominianni
Warshawsky
Ardecky
Paterniti
Tyhonas
Karanewsky
Kauffman
Broderick
Oldham
Montrose-Rafizadeh
Winneroski
Faul
McCarthy
Propionic acid derivative 8, which was designed and synthesized based on putative pharmacophores of known PPARγ- and PPARα-selective compounds, exhibits potent dual PPARα/γ agonist activity as demonstrated by in vitro binding and dose overlap in the newly
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