Journal of Medicinal Chemistry p. 5121 - 5124 (2003)
Update date:2022-08-04
Topics:
Xu, Yanping
Mayhugh, Daniel
Saeed, Ashraf
Wang, Xiaodong
Thompson, Richard C.
Dominianni, Samuel J.
Kauffman, Raymond F.
Singh, Jaipal
Bean, James S.
Bensch, William R.
Barr, Robert J.
Osborne, John
Montrose-Rafizadeh, Chahrzad
Zink, Richard W.
Yumibe, Nathan P.
Huang, Naijia
Luffer-Atlas, Debra
Rungta, Deepa
Maise, Dale E.
Mantlo, Nathan B.
A new series of hPPARα agonists containing a 2,4-dihydro-3H-1,2,4-triazol-3-one (triazolone) core is described leading to the discovery of 5 (LY518674), a highly potent and selective PPARα agonist.
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