Heterocyclic analogs of pleiadiene - XI. Synthesis of 1-(β-dialkylaminoalkyl)- and 2-aminoperimidines

Article abstract of DOI:10.1007/BF00472432

The corresponding 1-β-dialkylaminoethylperimidines were obtained by the action of β-dialkylaminoethyl chloride hydrochlorides on perimidines in alkaline media. Some of the compounds obtained form substituted 2-aminoperimidines and 2-perimidone on reaction with sodium amide or alkali. 2-Morpholino- and 2-piperidino-1-methylperimidines are obtained from 1-methyl-2-chloroperimidine and morpholine or piperidine. The synthesized compounds have weak bacteriostatic, fungistatic, and tuberculostatic activity.