Journal of Medicinal Chemistry p. 3483 - 3486 (2004)
Update date:2022-09-26
Topics:
Tucci, Fabio C.
Zhu, Yun-Fei
Guo, Zhiqiang
Gross, Timothy D.
Connors Jr., Patrick J.
Gao, Yinghong
Rowbottom, Martin W.
Struthers, R. Scott
Reinhart, Greg J.
Xie, Qiu
Chen, Ta Kung
Bozigian, Haig
Bonneville, Anne L. Killam
Fisher, Andrew
Jin, Liping
Saunders, John
Chen, Chen
Uracils possessing N-3 side chains derived from various amino alcohols were designed and synthesized as potent human gonadotropin releasing hormone receptor antagonists. The compounds herein presented displayed superior metabolic stability than their pred
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