Evidence of the Preferential Involvement of μ Receptors in Analgesia Using Enkephalins Highly Selective for Peripheral μ or δ Receptors

DOI: 10.1021/jm00142a002

Source and publish data:

Journal of Medicinal Chemistry p. 1119 - 1124 (1981)

Update date:2022-09-26

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Authors:

Gacel, Gilles

Fournie-Zaluski, Marie-Claude

Fellion, Etienne

Roques, Bernard P.

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Article abstract of DOI:10.1021/jm00142a002

In order to study the preferential involvement of μ or δ receptors in the analgesic effects of enkephalins, several peptides which selectively interact with these two kinds of receptors in peripheral organs were synthesized.The inhibitory potency on the e

Full text of DOI:10.1021/jm00142a002

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