Evidence of the Preferential Involvement of μ Receptors in Analgesia Using Enkephalins Highly Selective for Peripheral μ or δ Receptors

DOI: 10.1021/jm00142a002

Source and publish data:

Journal of Medicinal Chemistry p. 1119 - 1124 (1981)

Update date:2022-09-26

Topics:

Authors:

Gacel, Gilles

Fournie-Zaluski, Marie-Claude

Fellion, Etienne

Roques, Bernard P.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00142a002

In order to study the preferential involvement of μ or δ receptors in the analgesic effects of enkephalins, several peptides which selectively interact with these two kinds of receptors in peripheral organs were synthesized.The inhibitory potency on the e

Full text of DOI:10.1021/jm00142a002

Products guided by the article

Product name:N-(tert-butyloxycarbonyl)-L-tyrosyl-O-tert-butyl-D-serine methyl ester

Cas No:78537-13-0

R&D Labs maybe for 78537-13-0

Zhengzhou HQ Material Co.,Ltd

Contact:+86-371-67759225

Address:No.32, Jinsuo Road, High-tech Zone
Joyochem Co., Ltd.

website:https://sdjingyuan.lookchem.com/

Contact:86-531-82687998

Address:Factory Building 11, Jinan Comprehensive free trade zone, Shandong, China
Jinan Hongfangde Pharmatech Co.,Ltd

Contact:86-531-88870908

Address:F Bldg. West Unit North Area of Univ. Tech. Garden Xinyu Rd. Jinan New & High Tech Industry Development Zone Shandong, China
Shanghai Hohance Chemical Co., ltd

Contact:13914753421

Address:Fl.5；Bld. 70, Lane 1500; Xinfei Road
Goldwills Pharmaceuticals Co., Ltd.

Contact:0916-2237889 13991621155

Address:North Suburb of Hanzhong city, Shaanxi Province

Relevant to this article

USE OF 2-ETHOXY-1-ETHOXYCARBONYL-1,2-DIHYDROQUINOLINE AS CONDENSING AGENT IN THE SYNTHESIS OF FRAGMENT 20 - 24 OF THE SEQUENCE OF ACTH

Doi:10.1007/BF00579967
(1983)
Reaction of Organolithium Compounds with a Triphenylcyclopropyl Derivative. The Matter of Cyclopropyl Anion Ring Opening

Doi:10.1021/jo00335a063
(1981)
An Efficient Synthesis of Anhydroalditols and Allyl C-Glycosides

Doi:10.1021/jo00381a030
(1987)
Synthesis of 5-substituted-3-phenacyloxime-1,2,4-oxadiazoles from acetylated or benzoylated benzoylthiacetamide with hydroxylamine hydrochloride. Spectral evidence for a tetrahedral carbinolamine intermediate

Doi:10.1016/S0040-4020(01)92460-3
(1981)
Phase-transfer catalyzed alkylation and cycloalkylation of 3-substituted-1H-pyrazol-2-in-5-ones in the absence or presence of carbon disulphide

Doi:10.1080/104265090517208
(2005)
Synthesis of β-lactams from acetic acids and imines induced by phenyl dichlorophosphate reagent

Doi:10.1016/S0040-4020(01)96484-1
(1985)

Article Doi