RSC Medicinal Chemistry p. 665 - 675 (2020)
Update date:2022-08-05
Topics: Structural features Specificity
Bernasconi, Elena
Bertoni, Francesco
Caflisch, Amedeo
Cascione, Luciano
Dong, Jing
Gaudio, Eugenio
Jessen-Trefzer, Claudia
Nevado, Cristina
Pachmayr, Johanna
Sartori, Giulio
Spiliotopoulos, Dimitrios
Tarantelli, Chiara
Unzue, Andrea
Zahler, Stefan
Zhao, Hongtao
?led?, Pawe?
The X-ray structure of the catalytic domain of the EphA3 tyrosine kinase in complex with a previously reported type II inhibitor was used to design two novel quinoxaline derivatives, inspired by kinase inhibitors that have reached clinical development. Th
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