Synthesis and biological evaluation of phosphonamidate peptide inhibitors of enkephalinase and angiotensin-converting enzyme

DOI: 10.1021/jm00147a015

Source and publish data:

Journal of Medicinal Chemistry p. 1208 - 1216 (1985)

Update date:2022-07-30

Topics:

Authors:

Elliott Elliott

Marks Marks

Berg Berg

Portoghese

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00147a015

The effectiveness of phosphonamidate peptide analogues as inhibitors of rat kidney or human brain metallo-endopeptidase (enkephalinase, E.C. 3.4.24.11) and angiotensin-converting enzyme (ACE, 3.4.15.1) has been explored with a series of enkephalin analogu

Full text of DOI:10.1021/jm00147a015

Products guided by the article

Product name:CbzTyr(OBzl)-D-Ala

Cas No:96915-00-3

R&D Labs maybe for 96915-00-3

Borun Chemical Co.,Ltd.

Contact:+86-574- 87178138; 87297407

Address:No. 809, Liudingxingzuo, cangsong road, Ningbo, China
Cartoon Ingredients Co., Ltd

website:http://www.cartoonchem.com/

Contact:+86-25-58074918

Address:Room 2109, RuiHua Business Center,315 South ZhongShan Road, Nanjing 210001, China
Amadis Chemical Co., Ltd.

website:http://www.amadischem.com

Contact:86-571-89925085

Address:Watts Cosine.No.166.Xiangmao Road.
Chemvon Biotechnology Co. Ltd.

website:http://www.chemvon.com

Contact:86-21-58550039;86-21-31268550-8004

Address:Suite B-10#, 6999 Chuansha Road, Pudong District, Shanghai 201202, China
Lanzhou huibang biological chemical technology Co., LTD

Contact:0931-7843964

Address:NO.2011,Yannan Road,Chengguan,

Relevant to this article

Molecular Mechanism of Action of 5,6-Dihydroxytryptamine. Synthesis and Biological Evaluation of 4-Methyl-, 7-Methyl-, and 4,7-Dimethyl-5,6-dihydroxytryptamines

Doi:10.1021/jm00147a027
(1985)
Copper-catalyzed oxidative C-O bond formation of 2-acyl phenols and 1,3-dicarbonyl compounds with ethers: Direct access to phenol esters and enol esters

Doi:10.1021/jo500576x
(2014)
ADDITION REGIOSELECTIVE D'ORGANOMETALLIQUES α-INSATURES OU α-FONCTIONNELS AU CHLORURE DE N-ETHOXYCARBONYLPYRIDINIUM: SYNTHESE DE DIHYDRO-1,2 (OU-1,4)PYRIDINES 2-(OU-4)SUBSTITUTEES.

Doi:10.1016/S0040-4039(00)98503-4
(1985)
Lewis Acid Mediated Thienium Cation Diels-Alder Reaction: A New Method for Regio- and Stereoselective Functionalization of 1,3-Dienes

Doi:10.1016/S0040-4039(00)89135-2
(1985)
Cu(i) mediated Kinugasa reactions of α,β-unsaturated nitrones: A facile, diastereoselective route to 3-(hydroxy/bromo)methyl-1-aryl-4-(-styryl)azetidin-2-ones

Doi:10.1039/c6nj01747a
(2016)
Doi:10.1021/ja01520a067
(1959)

Article Doi