Synthesis and biological evaluation of phosphonamidate peptide inhibitors of enkephalinase and angiotensin-converting enzyme

DOI: 10.1021/jm00147a015

Source and publish data:

Journal of Medicinal Chemistry p. 1208 - 1216 (1985)

Update date:2022-07-30

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Authors:

Elliott Elliott

Marks Marks

Berg Berg

Portoghese

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Article abstract of DOI:10.1021/jm00147a015

The effectiveness of phosphonamidate peptide analogues as inhibitors of rat kidney or human brain metallo-endopeptidase (enkephalinase, E.C. 3.4.24.11) and angiotensin-converting enzyme (ACE, 3.4.15.1) has been explored with a series of enkephalin analogu

Full text of DOI:10.1021/jm00147a015

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