SYNTHESIS OF (E)-β-FLUOROMETHYLENEGLUTAMIC ACID

DOI: 10.1016/S0040-4039(00)89300-4

Source and publish data:

Tetrahedron Letters p. 4091 - 4092 (1985)

Update date:2022-08-05

Topics:

Authors:

McDonald, Ian A.

Palfreyman, Michael G.

Jung, Michel

Bey, Philippe

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Article abstract of DOI:10.1016/S0040-4039(00)89300-4

A potential dual-enzyme activated inhibitor of γ-aminobutyric acid transaminase, (E)-β-fluoromethyleneglutamic acid, was prepared from ethyl 3,3-dimethylacrylate in 11 steps.

Full text of DOI:10.1016/S0040-4039(00)89300-4

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