A selective protection of 2,3-diaminopropionic acid

Article abstract of DOI:10.1080/00397919308009829

A two step selective protection of 2,3-diaminopropionic acid yields the useful diaminopropionic acid methyl ester 3a. Further manipulation yields 2(S)-(N-benzyloxycarbonylamino)-3-aminopropionic acid methyl ester hydrochloride 5 in >99.9%ee.

Full text of DOI:10.1080/00397919308009829

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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A Selective Protection of 2,3-
Diaminopropionic Acid
a
a
M. S. Egbertson , C. F. Homnick & G. D. Hartman
a
a
Department of Medicinal, Chemistry Merck
Research Laboratories, West Point, PA. 19486
Version of record first published: 27 Oct 2006.
To cite this article: M. S. Egbertson , C. F. Homnick & G. D. Hartman (1993): A
Selective Protection of 2,3-Diaminopropionic Acid, Synthetic Communications: An
International Journal for Rapid Communication of Synthetic Organic Chemistry, 23:5,
703-709
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