
Journal of Medicinal Chemistry p. 4950 - 4952 (1995)
Update date:2022-08-17
Topics:
Thurkauf
Yuan
Chen
Wasley
Meade
Woodruff
Huston
Ross
A series of 1-phenyl-3-(aminomethyl)pyrroles were prepared in two steps from aniline and their affinities for D2, D3, and D4 dopamine receptor subtypes determined. A 15-fold selectivity for cloned human D4 recep
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