Novel applications of ethyl glyoxalate with the Ugi MCR

DOI: 10.1016/S0040-4039(99)00960-0

Source and publish data:

Tetrahedron Letters p. 5295 - 5299 (1999)

Update date:2022-08-29

Topics:

Authors:

Hulme, Christopher

Cherrier

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Article abstract of DOI:10.1016/S0040-4039(99)00960-0

This letter describes novel high-yielding solution phase preparations of 1,4-benzodiazepine-2,5-dione, diketopiperazine, ketopiperazine and dihydroquinoxalinone libraries via a UDC (Ugi/de-Boc/cyclization) strategy in combination with ethylglyoxalate. The

Full text of DOI:10.1016/S0040-4039(99)00960-0

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