Novel applications of ethyl glyoxalate with the Ugi MCR

DOI: 10.1016/S0040-4039(99)00960-0

Source and publish data:

Tetrahedron Letters p. 5295 - 5299 (1999)

Update date:2022-08-29

Topics:

Authors:

Hulme, Christopher

Cherrier

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(99)00960-0

This letter describes novel high-yielding solution phase preparations of 1,4-benzodiazepine-2,5-dione, diketopiperazine, ketopiperazine and dihydroquinoxalinone libraries via a UDC (Ugi/de-Boc/cyclization) strategy in combination with ethylglyoxalate. The

Full text of DOI:10.1016/S0040-4039(99)00960-0

Products guided by the article

Product name:Methyl anthranilate

Cas No:134-20-3

R&D Labs maybe for 134-20-3

Shanghai Sunway Pharmaceutical Technology Co.,Ltd.

Contact:+86-21-5161 3915

Address:Shanghai YangPu
ShangHai Original Economy-Trade Develop Co.,Ltd.,

Contact:86-21-68552131

Address:shanghai
Shanghai Sungo Technology Chemical Co., Ltd

Contact:0086-21-51385579

Address:Room2010, F/20, Tonghua Plaza, NO 345 Jinxiang Road, Jinqiao Export Processing Zone, Shanghai, 201206 P.R.CHINA
BrightGene Bio-Medical Technology Co., Ltd.

website:https://en.bright-gene.com/

Contact:+86-512-62551801

Address:Building C25 - C31, No. 218 Xinghu Road, Suzhou Industrial Park, Suzhou, Jiangsu, China.
LABTER PARMATECH(BEIJING)CO.,LTD

website:http://www.labter.com.cn/

Contact:+86-10-56330744

Address:NO.19,TIANRONG STREET,DAXING BIOMEDICIAL BASE ,ZHONGGUANCUN SCIENCE AND TECHNOLOGY PARK,BEIJING ,CHINA

Relevant to this article

Ruthenium-Catalyzed [3 + 2] Cycloaddition of 2H-Azirines with Alkynes: Access to Polysubstituted Pyrroles

Doi:10.1021/acs.joc.6b02322
(2016)
Visible light-induced aerobic oxidative cross-coupling of glycine esters with α-angelicalactone: a facile pathway to γ-lactams

Doi:10.1039/c8ob01844h
(2018)
Synthesis of novel C2 and C1 symmetric chiraphos derivatives and their application in palladium-catalyzed miyauramichael reaction

Doi:10.1246/cl.130375
(2013)
8-Endo cyclization of (alkoxycarbonyl)methyl radicals: Radical ways for preparation of eight-membered-ring lactones

Doi:10.1021/ja980908d
(1998)
Synthesis and crystal structure of 7-bromo-3,3-dibutyl-8-methoxy-5-phenyl-2,3-dihydrobenzo[b][1,4]thiazepin-4(5H)-one

Doi:10.1177/1747519820907877
(2020)
5-Arylamino-2-methyl-4,7-dioxobenzothiazoles as inhibitors of cyclin-dependent kinase 4 and cytotoxic agents

Doi:10.1016/S0960-894X(00)00014-7
(2000)

Article Doi