Bioorganic and Medicinal Chemistry Letters p. 5536 - 5540 (2010)
Update date:2022-08-17
Topics:
Tyagarajan, Sriram
Chakravarty, Prasun K.
Zhou, Bishan
Fisher, Michael H.
Wyvratt, Mathew J.
Lyons, Kathy
Klatt, Tracy
Li, Xiaohua
Kumar, Sanjeev
Williams, Brande
Felix, John
Priest, Birgit T.
Brochu, Richard M.
Warren, Vivien
Smith, McHardy
Garcia, Maria
Kaczorowski, Gregory J.
Martin, William J.
Abbadie, Catherine
McGowan, Erin
Jochnowitz, Nina
Parsons, William H.
Voltage-gated sodium channels have been shown to play a critical role in neuropathic pain. With a goal to develop potent peripherally active sodium channel blockers, a series of low molecular weight biaryl substituted imidazoles, oxazoles, and thiazole ca
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