Mendeleev Communications p. 495 - 497 (2021)
Update date:2022-08-11
Topics:
Bakulev, Vasiliy A.
Beryozkina, Tetyana V.
Eltsov, Oleg S.
Fan, Zhijin
Galieva, Nadezhda A.
Lubec, Gert
Saveliev, Dmitriy A.
Xing, Jihong
The reactions of N-(benz[d]oxazol-2-yl)- or N-(benzo[d]-thiazol-2-yl)-substituted carbothioamides with sulfonyl azides proceed as replacement of thioxo substituent by the sulfonylimino group to afford the corresponding N'-sulfonylated amidines. Acetic acid thioamides react smoothly upon boiling in ethanol, while for thioamides of trifluoroacetic and benzoic acids heating to 80–90 °C was required. Among hybrid molecules thus prepared, bacteriostatic-, bactericidal- and fungistatic-active against S. aureus and C. albicans representatives were found.
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Doi:10.1007/s11095-018-2414-5
(2018)Doi:10.1039/c39860001409
(1986)Doi:10.1021/ja00160a073
(1990)Doi:10.1039/b301734f
(2003)Doi:10.2174/092986711793979760
(2011)Doi:10.1002/cmdc.201700225
(2017)