Cyclisation of histidine containing peptides in the solid-phase by anchoring the imidazole ring to trityl resins

DOI: 10.1016/S0040-4039(98)02459-9

Source and publish data:

Tetrahedron Letters p. 809 - 812 (1999)

Update date:2022-08-11

Topics:

Authors:

Sabatino, Giuseppina

Chelli, Mario

Mazzucco, Silvia

Ginanneschi, Mauro

Papini, Anna Maria

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Article abstract of DOI:10.1016/S0040-4039(98)02459-9

Head-to-tail histidine containing cyclopeptides can be efficiently synthesised by a three-dimensional orthogonal solid-phase strategy (Fmoc/tBu/allyl) via anchoring the imidazole ring to trityl-resins. Furthermore, Fmoc-His(Trt-)-OAl can be a useful starting support for the preparation of diketopiperazine combinatorial libraries.

Full text of DOI:10.1016/S0040-4039(98)02459-9

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