114715-35-4

Basic information

• Product Name: (R)-1-BENZYL-3-MESYLOXY PYRROLIDINE
• Synonyms: 3-PYRROLIDINOL, 1-(PHENYLMETHYL)-METHANESULFONATE (ESTER), (R);(R)-1-BENZYL-3-MESYLOXY PYRROLIDINE;(R)-1-BENZYL-3-METHANESULFONYLOXYPYRROLIDINE;R-MSBHP
• CAS NO: 114715-35-4
• Molecular Formula: C₁₂H₁₇NO₃S
• Molecular Weight: 255.33
• Mol File: 114715-35-4.mol
• Article Data: 13

Chemical Properties

• Boiling Point: 398.6±31.0 °C(Predicted)
• Appearance: /
• Density: 1.25±0.1 g/cm3(Predicted)
• PKA: 7.35±0.40(Predicted)
• CAS DataBase Reference: (R)-1-BENZYL-3-MESYLOXY PYRROLIDINE(CAS DataBase Reference)
• NIST Chemistry Reference: (R)-1-BENZYL-3-MESYLOXY PYRROLIDINE(114715-35-4)
• EPA Substance Registry System: (R)-1-BENZYL-3-MESYLOXY PYRROLIDINE(114715-35-4)

Safety Data

• Hazardous Substances Data: 114715-35-4(Hazardous Substances Data)

Usage

General Description

(R)-1-Benzyl-3-mesyloxy pyrrolidine is a chemical compound that belongs to the class of pyrrolidine derivatives. It is an organic compound with a molecular formula of C13H17NO3S and a molecular weight of 271.34 g/mol. (R)-1-BENZYL-3-MESYLOXY PYRROLIDINE is commonly used as an intermediate in chemical synthesis, particularly in the production of pharmaceuticals and agrochemicals. Its structure includes a benzyl group and a mesyloxy group, which makes it a valuable precursor for the synthesis of various bioactive compounds. Additionally, (R)-1-Benzyl-3-mesyloxy pyrrolidine is an important chiral building block, meaning it contains a specific arrangement of atoms that can be useful in the production of enantiomerically pure compounds. Its versatile reactivity and chiral nature make it a valuable tool in the field of organic chemistry.

Upstream product

• 100-52-7 benzaldehyde 
• 159497-65-1 N,N-dibenzylasparaginic acid dibenzyl ester 
• 137428-32-1 (2S)-2-[bis(phenylmethyl)amino]-1,4-butanediol 
• 124-63-0 methanesulfonyl chloride 
• 101385-90-4 (R)-N-benzyl-3-hydroxypyrrolidine 

Downstream Products

• 159063-16-8 (S)-1-benzylpyrrolidine-3-carbonitrile 
• 216311-58-9 methyl (S)-(+)-1-(phenylmethyl)-3-pyrrolidinecarboxylate 
• 216311-66-9 (3R)-2-(1-Benzylpyrrolidin-3-yl)acetic acid 
• 216311-64-7 Ethyl (3R)-2-(1-benzylpyrrolidin-3-yl)acetate 
• 1212293-24-7 (S)-1-Benzyl-pyrrolidine-3-carboxylic acid; hydrochloride 
• 740833-39-0 C₁₄H₁₇N₃ 
• 188616-79-7 2-[4-[(3S)-1-(tert-butoxycarbonyl)-3-pyrrolidinyl]oxy]phenylacetic acid ethyl ester 
• 114636-34-9 (3S)-1-benzyl-3-<(R)-α-methoxy-α-(trifluoromethyl)-α-phenylacetamido>pyrrolidine 
• 114636-30-5 (S)-(-)-1-benzyl-3-acetylaminopyrrolidine 
• 114636-33-8 (R)-N-(1-benzylpyrrolidine-3-yl)acetamide 
• 114715-39-8 (R)-1-benzyl-3-aminopyrrolidine 
• 161659-80-9 (3S)-1-Benzylpyrrolidine-3-carboxylic acid 
• 131852-53-4 (S)-1-benzyl-3-(tert-butoxycarbonylamino)pyrrolidine 
• 114715-38-7 (3S)-1-benzyl-3-pyrrolidinamine 

Relevant articles and documents

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Efficient synthesis of the 5-HT2C receptor agonist, Org 37684

An efficient synthesis of the 5-HT2C receptor agonist Org 37684 is presented. The synthesis utilises the regioselective demethylation of an arylether as the key step.